CPD-2828
CPD-2828 is an orally active and selective IRE1α inhibitor with an IC50 value of 1.2 μM. CPD-2828 is promising for research of endoplasmic reticulum stress-related diseases (e.g., cancer, neurodegenerative diseases).
For research use only. We do not sell to patients.
- Formula: C29H29N3O7
- Molecular Weight:531.56
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Protocols
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
IC50 & Target
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IRE1α 1.2 μM (IC50) |
Chemical Information
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Molecular Weight 531.56
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Formula C29H29N3O7
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SMILES
O=CC1=C(O)C=CC2=C1OC(C(CC(N3CCC(C4=CC=C(NC(CC5)C(NC5=O)=O)C=C4)CC3)=O)=C2C)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Protocols
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Cell Cytotoxicity Assay
Cytotoxicity assays are usually based on the assessment of cell membrane damage, which can also be indirectly detected by measuring cell viability. Detection methods include MTT assay, CKK-8 assay, LDH assay and ATP assay, etc.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CPD-2828 Related Classifications
HY-174991 Related Classifications
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