EGFR/PI3Kα-IN-1
EGFR/PI3Kα-IN-1 (compound 30k) is a dual EGFR/PI3Kα inhibitor with IC50 values of 3.6 nM (EGFRL858R/T790M) and 30 nM (PI3Kα), respectively. EGFR/PI3Kα-IN-1 can inhibit tumor cell proliferation and has anticancer activity.
For research use only. We do not sell to patients.
- Formula: C50H49N11O5S
- Molecular Weight:916.06
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
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Biological Activity
IC50: 3.6 nM (EGFRL858R/T790M); 30 nM (PI3Kα)[1]
Chemical Information
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Molecular Weight 916.06
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Formula C50H49N11O5S
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SMILES
NC1=CC2=C(O1)C=CC(C(C=C3)=CN4C3=NC=C4C(N5CCN(C(CCCCN6CCN(C7=CC=C(NC8=NC(C=CS9)=C9C(OC%10=CC(NC(C=C)=O)=CC=C%10)=N8)C=C7)CC6)=O)CC5)=O)=C2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
EGFR/PI3Kα-IN-1 Related Classifications
HY-161968 Related Classifications
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