Elenestinib phosphate
Elenestinib (BLU-263) phosphate is an orally active inhibitor of Tyrosine kinase with an IC50 of 0.2 nM for KIT D816V. Elenestinib phosphate minimally penetrates the blood-brain barrier. Elenestinib phosphate can be used in the study of systemic mastocytosis.
For research use only. We do not sell to patients.
- CAS No.: 2832013-93-9
- Formula: C27H32FN10O5P
- Molecular Weight:626.58
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
IC50: 0.2 nM (KIT D816V)[1]
Chemical Information
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CAS No. 2832013-93-9
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Molecular Weight 626.58
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Formula C27H32FN10O5P
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SMILES
OCCN1C=C(C=N1)C2=CN3N=CN=C(N4CCN(C5=NC=C([C@@](N)(C6=CC=C(C=C6)F)C)C=N5)CC4)C3=C2.OP(O)(O)=O
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Synonyms
BLU-263 phosphate
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)