Estrogen receptor β/HDAC probe 1
Estrogen receptor β/HDAC probe 1 (compound P1) is a near-infrared fluorescent probe that dual-targets the estrogen receptor (Estrogen Receptor/ERR) β/histone deacetylase HDAC.
For research use only. We do not sell to patients.
- CAS No.: 3057270-84-2
- Formula: C28H26N4O5
- Molecular Weight:498.53
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
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Help & FAQs
Biological Activity
Estrogen Receptor/ERR β[1]
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| DU-145 | IC50 |
0.96 μM
Compound: P1
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Antiproliferative activity against human DU-145 cells assessed as inhibition of cell growth incubated for 3 to 5 days by CCK-8 assay
Antiproliferative activity against human DU-145 cells assessed as inhibition of cell growth incubated for 3 to 5 days by CCK-8 assay
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[PMID: 38367494] |
| Vero | IC50 |
6.13 μM
Compound: P1
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Antiproliferative activity against green monkey Vero cells assessed as inhibition of cell growth incubated for 3 to 5 days by CCK-8 assay
Antiproliferative activity against green monkey Vero cells assessed as inhibition of cell growth incubated for 3 to 5 days by CCK-8 assay
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[PMID: 38367494] |
Chemical Information
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CAS No. 3057270-84-2
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Molecular Weight 498.53
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Formula C28H26N4O5
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SMILES
OC(C=C1)=C(NC(CCCCCCC(NO)=O)=O)C=C1/C=C/C2=C/C(C3=CC=CC=C3O2)=C(C#N)/C#N
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Estrogen receptor β/HDAC probe 1 Related Classifications
HY-D2280 Related Classifications
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