CB2R probe 1
CB2R probe 1 is a safe and green CB2R (cannabinoid 2 receptor) fluorescent probe with an Ki of 130 nM. CB2R probe 1 shows low cytotoxicity in cancer cells.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 2634714-79-5
- Fòrmula: C36H42N4O4
- Peso molecular:594.74
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Actividad biológica
Descripciòn
IC50 & Target
[1]|
cannabinoid type-2 receptors 130 nM (Ki) |
In Vitro
CB2R probe 1 (compound 28) (100 nM; 24 h) shows low cytotoxicity with IC50s of 1.6, 1.4, 1.4, 1.1, 2.6, 0.55, 2.0, 2.4, 2.8 nM for PANC1, U2OS, HT29, HT29-DX, U87AD, PC3, CB2R-HEK293, MCF7, MCFT-DX cells, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 2634714-79-5
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Peso molecular 594.74
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Fòrmula C36H42N4O4
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SMILES
CN(C1=CC2=C(C(N(C2=O)CCCCCCN3C=C(C(C4=CC=CC=C43)=O)C(N[C@@]5(CC6C7)CC7CC(C6)C5)=O)=O)C=C1)C
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)