country

Change Language

EN - English
FR - Français
DE - Deutsch
ES - Español
JA - 日本語
KO - 한국어

Country or Region:

United States

Product Name	Size / Unit Price	Qty

Total: USD 0.00 Checkout

Referencia número: HY-19241

Copy Link Print Information

CP-85958

CP-85958 is a specific leukotriene D₄ (LTD₄) receptor antagonist. CP-85958 can be used in the research of inflammatory diseases such as asthma.

Para uso exclusivo en investigación. No vendemos a pacientes.

No. CAS: 134002-60-1
Fòrmula: C₂₅H₂₀FNO₅S
Peso molecular:465.49

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (264 KB)

CP-85958 Chemical Structure

No. CAS: 134002-60-1

Tamaño

Precio

Stock

Cantidad

Amount: USD 0.00

* Seleccione Cantidad antes de agregar artículos.

Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Actividad biológica
- Descripciòn
- IC₅₀ & Target
- Cellular Effect
Chemical Information
Pureza y Documentación
Referencias
Calculators
Help & FAQs
Classifications
Bioz

Actividad biológica

Descripciòn

CP-85958 is a specific leukotriene D₄ (LTD₄) receptor antagonist. CP-85958 can be used in the research of inflammatory diseases such as asthma^[1].

IC₅₀ & Target

^[1]

LTD₄

Ver todos los productos específicos de isoformas Leukotriene Receptor :

Cellular Effect

Cell Line	Type	Value	Description	References
RBL-1	IC₅₀	8.1 μM Compound: 5 ((+)-CP-85958)	Inhibition of 5-Lipoxygenase (5-LO) in rat basophilic leukemia cells Inhibition of 5-Lipoxygenase (5-LO) in rat basophilic leukemia cells	10.1016/0960-894X(95)00225-I
U-937	IC₅₀	0.31 μM Compound: 3	Compound was evaluated for influx of calcium mobilization in human U937 cells Compound was evaluated for influx of calcium mobilization in human U937 cells	[PMID: 9873435]
U-937	IC₅₀	0.31 μM Compound: 3	Compound was tested for its ability to inhibit calcium influx in human U937 cells Compound was tested for its ability to inhibit calcium influx in human U937 cells	[PMID: 9934474]

Chemical Information

No. CAS 134002-60-1
Peso molecular 465.49
Fòrmula C₂₅H₂₀FNO₅S
SMILES

O=C(O)C1=CC=CC(C[C@@H]2COC3=CC=C(OCC4=NC5=CC(F)=CC=C5S4)C=C3[C@@H]2O)=C1
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureza y Documentación

Select Batch:

Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (264 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Marfat A, et al. The discovery of CP-96,021 and CP-96,486, balanced, combined, potent and orally active leukotriene D4 (LTD4)/platelet activating factor (PAF) receptor antagonists. Bioorganic & Medicinal Chemistry Letters, 1995, 5(13): 1377-1382.

Calculators

Calculadora de molaridad

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculadora de dilución

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

Keywords

MOQ

Minimum order quantity

100 mg

Obtener un presupuesto En stock

Other size

Obtener un presupuesto

Amount: USD 0.00

Actividad biológica
- Descripciòn
- IC₅₀ & Target
Chemical Information
Pureza y Documentación
Referencias

Nombre del producto:
Referencia número:
Cantidad:
MCE Japan Authorized Agent:

Nombre del producto:
No. CAS:
Species:
Pureza:
Cantidad:

CP-85958

Ver todos los productos específicos de isoformas Leukotriene Receptor

Actividad biológica

Descripciòn

IC50 & Target

Cellular Effect

Chemical Information

Pureza y Documentación

Referencias

Calculators

Help & FAQs

CP-85958 Related Classifications

HY-19241 Related Classifications

Bioz

Keywords

Your Recently Viewed Products

IC₅₀ & Target