PV1115
PV1115 is a potent and highly selective Chk2 inhibitor with an IC50 of 0.14 nM, 66000 nM, >100000 nM for Chk2, Chk1 and RSK2, respectively. PV1115 is situated within the ATP-binding pocket of Chk2.
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- No. CAS: 1093793-10-2
- Fòrmula: C20H19N7O3
- Peso molecular:405.41
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Actividad biológica
IC50: 0.14 nM (Chk2), 66000 nM (Chk1) and >100000 nM (RSK2)[1]
Chemical Information
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No. CAS 1093793-10-2
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Peso molecular 405.41
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Fòrmula C20H19N7O3
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SMILES
O=C(NC1=CC=C(C=C1)/C(C)=N/NC2=NCCN2)C3=CC4=C(C([N+]([O-])=O)=CC=C4)N3
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)