H4R antagonist 2
Based on 1 Customer Validation
H4R antagonist 2 (page 68), a Furo[3,2-d]pyrimidine derivative, is a potent H4R antagonist. H4R antagonist 2 can be used in research of rheumatoid arthritis.
For research use only. We do not sell to patients.
- Purity: 98.92%
- CAS No.: 1148115-99-4
- Formula: C13H17N5O
- Molecular Weight:259.31
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Storage:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
All Histamine Receptor Isoforms
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Biological Activity
Chemical Information
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CAS No. 1148115-99-4
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Appearance Solid
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Molecular Weight 259.31
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Formula C13H17N5O
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Color White to yellow
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SMILES
NC1=NC(N2CC(NC)C2)=C(OC3=C4CCC3)C4=N1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : 15 mg/mL (57.85 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (273 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 3.8564 mL | 19.2819 mL | 38.5639 mL | 96.4097 mL |
| 5 mM | 0.7713 mL | 3.8564 mL | 7.7128 mL | 19.2819 mL | |
| 10 mM | 0.3856 mL | 1.9282 mL | 3.8564 mL | 9.6410 mL | |
| 15 mM | 0.2571 mL | 1.2855 mL | 2.5709 mL | 6.4273 mL | |
| 20 mM | 0.1928 mL | 0.9641 mL | 1.9282 mL | 4.8205 mL | |
| 25 mM | 0.1543 mL | 0.7713 mL | 1.5426 mL | 3.8564 mL | |
| 30 mM | 0.1285 mL | 0.6427 mL | 1.2855 mL | 3.2137 mL | |
| 40 mM | 0.0964 mL | 0.4820 mL | 0.9641 mL | 2.4102 mL | |
| 50 mM | 0.0771 mL | 0.3856 mL | 0.7713 mL | 1.9282 mL |