1. Metabolic Enzyme/Protease
  2. Isocitrate Dehydrogenase (IDH)
  3. IDH1 Inhibitor 2

IDH1 Inhibitor 2 

Cat. No.: HY-128661
Handling Instructions

IDH1 Inhibitor 2 is a potent IDH1 inhibitor via a direct covalent modification of His315, with an IC50 of 110 nM.

For research use only. We do not sell to patients.

IDH1 Inhibitor 2 Chemical Structure

IDH1 Inhibitor 2 Chemical Structure

CAS No. : 2244895-42-7

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Description

IDH1 Inhibitor 2 is a potent IDH1 inhibitor via a direct covalent modification of His315, with an IC50 of 110 nM[1].

IC50 & Target

IC50: 110 nM (IDH1)[1].

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
Molecular Weight

406.48

Formula

C₂₆H₂₂N₄O

CAS No.

2244895-42-7

SMILES

N#CC1=C[[email protected]@]2(C3=CC=CC=C3)[[email protected]](CCC4=C2N=C(NC5=CC=CC=C5)N=C4)([H])[[email protected]](C)C1=O

Shipping

Room temperature in continental US; may vary elsewhere

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  • Dilution Calculator

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
IDH1 Inhibitor 2
Cat. No.:
HY-128661
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IDH1 Inhibitor 2

Cat. No.: HY-128661