Pegcantratinib
Pegcantratinib (CT327) is a potent and selective TRKA antagonist with activity against TRKB and TRKC. Pegcantratinib can be used for research of CYLD cutaneous syndrome (CCS) and inflammatory dermatoses, such as psoriasis and concomitant pruritus.
For research use only. We do not sell to patients.
- CAS No.: 1233363-33-1
- Formula: (C2H4O)nC30H24N4O6
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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TrkA |
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 1233363-33-1
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Formula (C2H4O)nC30H24N4O6
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SMILES
O=C(N(CCOCCCOCC)C(O1)=O)[C@@]21[C@](C)(O3)N(C4=CC=CC=C45)C6=C5C7=C(C(NC7)=O)C8=C6N([C@H]3C2)C9=CC=CC=C98.[n]
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Synonyms
CT327; SNA-120
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)