VA-111913
VA-111913 (VT-913) is a vasopressin receptor V1A antagonist (Ki = 1.74 nM). VA-111913 reduces uterine contractions and improves uterine blood flow by inhibiting vasopressin, thereby alleviating dysmenorrhea. VA-111913 can be used for research on menstrual pain.
For research use only. We do not sell to patients.
- CAS No.: 877856-17-2
- Formula: C23H21ClFN5O2
- Molecular Weight:453.90
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Vasopressin Receptor Isoforms
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Biological Activity
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V1a Receptor 1.74 nM (Ki) |
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 877856-17-2
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Molecular Weight 453.90
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Formula C23H21ClFN5O2
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SMILES
O=C(C1CC1)NCC2=CC=C(C(N3CC4=C(N(C)N=C4)NC5=CC(Cl)=CC=C35)=O)C=C2F
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Synonyms
VT-913
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)