VU6036864
VU6036864 (compound 45) is an orally active, selective mAChR M5 antagonist with IC50=20 nM for human M5. VU6036864 is >500-fold selective for human M1-4, with BBB characteristic and high oral bioavailability (%F>100%).
For research use only. We do not sell to patients.
- CAS No.: 2746406-36-8
- Formula: C15H12D4ClN5O3S
- Molecular Weight:385.86
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
IC50: 20 nM (human mAChR M5)[1]
1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.
Chemical Information
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CAS No. 2746406-36-8
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Unlabeled Cas 2746405-41-2
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Molecular Weight 385.86
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Formula C15H12D4ClN5O3S
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SMILES
CC1=NC=C(S(=O)(N2C([2H])([2H])CC(C3=CN4C(C=C3Cl)=NC=N4)CC2([2H])[2H])=O)O1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
VU6036864 Related Classifications
HY-159578S Related Classifications
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