PAT-IN-1
PAT-IN-1 is a protein acyl transferases (PAT) inhibitor. PAT-IN-1 competitively inhibits Erf2 autopalmitoylation (WO2017011518A1; compound 13).
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- CAS 番号: 2066571-97-7
- 分子式: C45H68N4O
- 分子量:681.05
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
生物活性
製品説明
体外実験
PAT-IN-1 (compound 13) completely inhibits growth of RJY1941 (control) at 20 μΜ, but has no detectable effect at lower concentrations. PAT-IN-1 inhibits (100%) the growth of RJY1942 (palmitoylation sensitive) at 5 μΜ[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 2066571-97-7
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分子量 681.05
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分子式 C45H68N4O
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SMILES
CC(C1=CC=C(C=C1)CC(C)C)CN(CCN(C2)CCCC[C@@H]3N(CCNC3)CC(C4=CC=C(C=C4)CC(C)C)C)[C@H]2CC5=CC=C(C=C5)O
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
ホットトピック
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Topics
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Topics Palmitoylation: Bridging Physiology and Disease
Palmitoylation is a reversible lipid modification in which palmitate is covalently attached to protein cysteine residues, thereby regulating protein localization, stability, membrane association, and signaling activity.
2026-06-18
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)