PREP-IN-2
PREP-IN-2 is an irreversible and selective prolyl endopeptidase (PREP) inhibitor with an IC50 of 0.53 μM and a Ki of 0.62 μM. PREP-IN-2 can be used in research related to neurodegenerative diseases and triple-negative breast cancer.
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研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 分子式: C22H24ClN5O2
- 分子量:425.91
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
生物活性
PREP-IN-2 (Compound 14) (0.001-10 μM; 4 h) inhibits PREP activity in SH-SY5Y and MDA-MB-231 cells, with IC50 values of 67 nM and 127 nM, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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分子量 425.91
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分子式 C22H24ClN5O2
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SMILES
ClC1=C(C(NCC(N2CCCC2)=O)=O)C=NC3=C1C(C)=NN3CCC4=CC=CC=C4
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)