LEI-101 free base
LEI-101 free base is a selective and orally bioavailable CB2 receptor agonist with the potential to inhibit diseases associated with inflammation and/or oxidative stress. LEI-101 free base has a binding potency to CB2 receptors that is approximately 100 times higher than that to CB1 receptors. Its pEC50 value on CB2 receptors is 8, while its pKi value on hERG is less than 4. LEI-101 may have an inhibitory effect on conditions such as kidney disease.
For research use only. We do not sell to patients.
- CAS No.: 1228660-00-1
- Formula: C23H25FN4O4S
- Molecular Weight:472.53
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Endogenous Metabolite Isoforms
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Biological Activity
Chemical Information
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CAS No. 1228660-00-1
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Molecular Weight 472.53
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Formula C23H25FN4O4S
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SMILES
O=C1N(C(CN1CC2=CC=C(C=C2)C3=NC(CN(CC4)CCS4(=O)=O)=C(C=C3)F)=O)C5CC5
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)