LSD1-IN-22
LSD1-IN-22 is a potent Lysine-specific demethylase 1 (LSD1) inhibitor with a Ki value of 98 nM. LSD1-IN-22 has anti-proliferative activity against certain cancer cells.
For research use only. We do not sell to patients.
- CAS No.: 2821068-05-5
- Formula: C9H8BrF2N
- Molecular Weight:248.07
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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KDM1/LSD1 |
LSD1-IN-22 (compound 7t) has anti-proliferative activity against CCRF-CEM, Jurkat and hERG cells[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
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Cell Line:CCRF-CEM, Jurkat and hERG
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Concentration:0-50 μM
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Incubation Time:72 h
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Result:Exhibited anti-proliferative activity against CCRF-CEM, Jurkat and hERG cells with IC50s of 23±0.8 μM, 26±1.7 μM and 7.7±1.3 μM.
Chemical Information
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CAS No. 2821068-05-5
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Molecular Weight 248.07
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Formula C9H8BrF2N
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SMILES
N[C@H]1[C@H](C2=CC(F)=C(Br)C=C2F)C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)