Lu 26-046
Lu 26-046 is the agonist for muscarinic M1 receptor and M2 receptor and a weak antagonist for M3 receptor, with Ki of 0.51, 26 and 5 nM, respectively. Lu 26-046 exhibits specific stimulus property, that can be recognized by rats.
For research use only. We do not sell to patients.
- CAS No.: 143756-51-8
- Formula: C10H12N2OS
- Molecular Weight:208.28
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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mAChR1 0.51 nM (Ki) |
mAChR3 5 nM (Ki) |
mAChR2 26 nM (Ki) |
Chemical Information
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CAS No. 143756-51-8
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Molecular Weight 208.28
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Formula C10H12N2OS
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SMILES
C#CCOC1=NSC2=C1CNC[C@H]2C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)