MAGL-IN-9
MAGL-IN-9 (compound 16) is a selective and reversible MAGL inhibitor with IC50 2.7 nM.
For research use only. We do not sell to patients.
- CAS No.: 3017151-74-2
- Formula: C25H22F4N2O2S
- Molecular Weight:490.51
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
IC50: 2.7 nM (MAGL)[1]
MAGL-IN-9 (10 μM, 25 min) selectively inhibits MAGL in mouse brain membrane preparations, without affecting other serine hydrolases such as FAAH, ABHD6, and ABHD12[1].
MAGL-IN-9 shows a reversible inhibition mechanism in both preincubation and dilution tests[1].
MAGL-IN-9 inhibits MAGL in U973 cells with an IC50 value of 193 nM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3017151-74-2
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Molecular Weight 490.51
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Formula C25H22F4N2O2S
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SMILES
O=C(N1CCC(CC2=CC=C(F)C(SC3=NC=CC(C(F)(F)F)=C3)=C2)CC1)C4=CC=CC(O)=C4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
MAGL-IN-9 Related Classifications
HY-157040 Related Classifications
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