PI3Kδ/BET-IN-1
PI3Kδ/BET-IN-1 (compound 10b) shows excellent and balanced activities against PI3Kδ (IC50 = 112 nM) and BRD4-BD1 (IC50 = 19 nM) and exhibits strong antiproliferative activities in DLBCL cells.
연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.
- CAS No.: 3054869-10-9
- 화학식: C27H34N6O3S
- 분자량:522.66
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보관:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
|
PI3Kδ 112 nM (IC50) |
BRD4 (BD1) 19 nM (IC50) |
Chemical Information
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CAS No. 3054869-10-9
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분자량 522.66
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화학식 C27H34N6O3S
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SMILES
CN1C=C(C2=NC(N3CCOCC3)=C4SC(CN5CCC(C(C)(O)C)CC5)=CC4=N2)C6=C(C1=O)NC=C6
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)