PI3Kδ/BET-IN-1
PI3Kδ/BET-IN-1 (compound 10b) shows excellent and balanced activities against PI3Kδ (IC50 = 112 nM) and BRD4-BD1 (IC50 = 19 nM) and exhibits strong antiproliferative activities in DLBCL cells.
For research use only. We do not sell to patients.
- CAS No.: 3054869-10-9
- Formula: C27H34N6O3S
- Molecular Weight:522.66
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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PI3Kδ 112 nM (IC50) |
BRD4 (BD1) 19 nM (IC50) |
Chemical Information
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CAS No. 3054869-10-9
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Molecular Weight 522.66
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Formula C27H34N6O3S
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SMILES
CN1C=C(C2=NC(N3CCOCC3)=C4SC(CN5CCC(C(C)(O)C)CC5)=CC4=N2)C6=C(C1=O)NC=C6
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
PI3Kδ/BET-IN-1 Related Classifications
HY-172130 Related Classifications
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