Bis(heteroaryl)piperazine (BHAP) reverse transcriptase inhibitors: structure-activity relationships of novel substituted indole analogues and the identification of 1-[(5-methanesulfonamido-1H-indol-2-yl)-carbonyl]-4-[3- [(1-methylethyl)amino]-pyridinyl]piperazine monomethanesulfonate (U-90152S), a second-generation clinical candidate

  • J Med Chem. 1993 May 14;36(10):1505-8. doi: 10.1021/jm00062a027.
D L Romero  1 ,  R A Morge ,  M J Genin ,  C Biles ,  M Busso ,  L Resnick ,  I W Althaus ,  F Reusser ,  R C Thomas ,  W G Tarpley
Affiliations
  • 1. Upjohn Laboratories, Kalamazoo, Michigan 49001.
PMID: 7684450 DOI: 10.1021/jm00062a027