Pynazolam
Pynazolam is a predicted positive allosteric modulator of GABAA receptor. 3D-field QSAR and RVM models predict an IC50 of approximately 0.40 nM. Pynazolam can be used in studies related to GABAA receptor pharmacology.
For research use only. We do not sell to patients.
- CAS No.: 2034366-97-5
- Formula: C16H12N6O2
- Molecular Weight:320.31
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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GABAA receptor |
Pynazolam is predicted to be one of the most active designer benzodiazepines at the GABA-AR, with a log 1/c value of 9.4, indicating potent inhibitory activity in displacing [3H]-diazepam from rat cerebral cortex binding sites[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2034366-97-5
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Molecular Weight 320.31
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Formula C16H12N6O2
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SMILES
O=[N+](C1=CC=C(N2C(CN=C3C4=NC=CC=C4)=NN=C2C)C3=C1)[O-]
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)