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(R,R)-Birelentinib

(Synonyms: (R,R)-DZD8586)

(R,R)-Birelentinib ((R,R)-DZD8586) (Compound 14) is a potent BTK inhibitor with IC50 values for BTK WT and BTK C481S of 0.7 and 0.86 nM, respectively. (R,R)-Birelentinib inhibits the self-phosphorylation of BTK and its IC50 is 24.3 nM. (R,R)-Birelentinib exhibits significant anti-proliferative activity against wild-type and C481S mutant HEK293 cells. (R,R)-Birelentinib can be used for the study of drug-resistant B-cell malignancies.

For research use only. We do not sell to patients.

  • CAS No.: 2662512-14-1
  • Formula: C23H21F2N5O3
  • Molecular Weight:453.45
  • Storage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

  • (R,R)-Birelentinib Chemical Structure
    (R,R)-Birelentinib Chemical Structure
CAS No.: 2662512-14-1
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  • (R,R)-Birelentinib Chemical Structure
    (R,R)-Birelentinib Chemical Structure
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  • (R,R)-Birelentinib