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Cat. No.: HY-151805

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RGT-068A

RGT-068A is a MALT1 inhibitor with oral bioavailability. RGT-068A inhibits MALT1 activity. RGT-068A can be used for the research of autoimmune diseases.

For research use only. We do not sell to patients.

CAS No.: 2577171-33-4
Formula: C₁₇H₁₆ClN₉O₂
Molecular Weight:413.82

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (269 KB)

RGT-068A Chemical Structure

CAS No.: 2577171-33-4

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
- In Vivo
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Bioz

Biological Activity

Description

RGT-068A is a MALT1 inhibitor with oral bioavailability. RGT-068A inhibits MALT1 activity. RGT-068A can be used for the research of autoimmune diseases^[1].

IC₅₀ & Target

MALT1^[1]

In Vivo

RGT-068A exhibits favorable oral bioavailability^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 2577171-33-4
Molecular Weight 413.82
Formula C₁₇H₁₆ClN₉O₂
SMILES

CO[C@H](C1=C(C=NN2C=CN=C12)NC(NC3=CN=C(C(Cl)=C3)N4N=CC=N4)=O)C
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (269 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Feng S, et al. Direct Construction of Chiral Ether via Highly Efficient Heck Reaction and N-Directed Asymmetric Hydrogenation for Large-Scale Synthesis of MALT1 Inhibitor RGT-068A. Organic Process Research & Development. 2022 Nov 3;26(11):3089-95.

Calculators

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Dilution Calculator

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

100 mg

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