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Cat. No.: HY-175256

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RSK2-IN-5

RSK2-IN-5 (compoud C24) is a p90 ribosomal S6 kinase 2 (RSK2) inhibitor with a K_d of 317 nM. RSK2-IN-5 exhibits antitumor activity against breast cancer and melanoma cancer cells.

For research use only. We do not sell to patients.

Purity: 90.0%
CAS No.: 799832-19-2
Formula: C₂₄H₂₅N₅O₂
Molecular Weight:415.49

Storage:

Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month

RSK2-IN-5 Chemical Structure

CAS No.: 799832-19-2

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

RSK2-IN-5 (compoud C24) is a p90 ribosomal S6 kinase 2 (RSK2) inhibitor with a K_d of 317 nM. RSK2-IN-5 exhibits antitumor activity against breast cancer and melanoma cancer cells^[1].

All Ribosomal S6 Kinase (RSK) Isoforms :

Chemical Information

CAS No. 799832-19-2
Appearance Solid
Molecular Weight 415.49
Formula C₂₄H₂₅N₅O₂
Color Light yellow to yellow
SMILES

O=C(C1=C(N)N(CC2=C(OC)C=CC=C2)C3=C1N=C4C=CC=CC4=N3)NC5CCCC5
Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Powder	-20°C	3 years
In solvent	-80°C	6 months
	-20°C	1 month

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (272 KB)
SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Yue Zhao, et al. Discovery of novel p90 ribosomal S6 kinase 2 inhibitors for potential cancer treatment through ligand-based and structure-based virtual screening methods. Chemometrics and Intelligent Laboratory Systems. Volume 217, 15 October 2021, 104402

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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RSK2-IN-5

All Ribosomal S6 Kinase (RSK) Isoforms

Biological Activity

Chemical Information

Purity & Documentation

References

Calculators

Help & FAQs

RSK2-IN-5 Related Classifications

HY-175256 Related Classifications