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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
369 Results for "
CI
" in MedChemExpress (MCE) Product Catalog:
Products (369)
369 Results for "CI" in MCE Product Catalog:
Cat. No.: HY-105504
CAS No.: 130116-16-4
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CI-986 is a dual inhibitor of COX and 5-LOX. CI-986 can prevent the coronary vasoconstriction and the increased production of LTB(4) and LTC(4). CI-986 also has anti-inflammatory and analgesic effects. CI-986 can be used for the researches of inflammation and cardiovascular disease, such as arthritis .
Cat. No.: HY-W516943
CAS No.: 700-07-2
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CI-624 decrease secretion volumes and outputs of hydrogen, sodium and potassium ions and of pepsin. CI-624 can be used in the research of cancer and autoimmune diseases .
Cat. No.: HY-146364
CAS No.: 2132412-25-8
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Cat. No.: HY-19108
CAS No.: 104795-68-8
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CI-959 is an orally active cell activation inhibitor. CI-959 selectively suppresses inflammatory cell activation post-receptor signaling via inhibiting calcium influx and weak calmodulin antagonism, without targeting PLC, PKC or NADPH oxidase. CI-959 blocks lung allergic mediator release, anti-IgE bronchial contraction, neutrophil function, T-cell proliferation and DC marker expression while sparing monocytes. CI-959 provides gastric cytoprotection by inhibiting leukocyte adhesion and suppresses tumor motility through F-actin reduction. CI-959 can be used for research on allergies, inflammation, autoimmune diseases, gastric injury, and tumor metastasis .
Cat. No.: HY-106752
CAS No.: 98383-40-5
Synonyms: MRS-3310
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CI-936 (MRS-3310) is an orally active A2 agonist with 25 nM affinity. CI-936 produces potent and selective effects in preclinical tests predictive of antipsychotic efficacy. CI-936 inhibits exploratory activity in mice .
Cat. No.: HY-123240
CAS No.: 110283-79-9
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CI-966 is a potent, selective, orally active and brain-penetrant inhibitor of the GABA transporter GAT-1, with IC50s of 0.26 μM and 1.2 μM for hGAT-1, rGAT-1, respectively. CI-966 shows more than 200-fold selectivity over GAT-2, GAT-3, and BGT-3. CI-966 exhibits anticonvulsant and neuroprotective activities .
Cat. No.: HY-105628A
CAS No.: 3734-16-5
Synonyms: CI-427 hydrochloride
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Prodilidine (CI-427) hydrochloride is a potent analgetic agent .
Cat. No.: HY-105226B
Synonyms: PD134308 hemihydrate
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CI-988 hemihydrate (PD134308) is a potent, selective and orally active CCK2R (cholecystokinin 2 receptor) antagonist with an IC50 of 1.7 nM for mouse cortex CCK2. CI-988 hemihydrate shows >1600-fold selectivity for CCK2 over CCK1 receptor. CI-988 hemihydrate has anxiolytic and anti-tumor effects .
Cat. No.: HY-119795
CAS No.: 51022-73-2
Synonyms: CI-781
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Zometapine (CI-781) is a pyrazolodiazepine derivative. Zometapine can be used in antidepressant research .
Cat. No.: HY-103459
CAS No.: 162256-50-0
Synonyms: PD156707
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CI-1020 (PD156707) is an orally active and selective antagonist targeting endothelin (ETA) with an IC50 value of 0.3 nM. CI-1020 blocks intimal hyperplasia in human saphenous veins completely in organ culture. CI 1020 inhibits hypoxic pulmonary hypertension and blocks ET-1-induced pressor responses following oral administration .
Cat. No.: HY-50295R
CAS No.: 212631-79-3
Synonyms: PD 184352 (Standard)
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CI-1040 (Standard) is the analytical standard of CI-1040. This product is intended for research and analytical applications. CI-1040 (PD 184352) is an orally active, highly specific, small-molecule inhibitor of MEK with an IC50 of 17 nM for MEK1.
Cat. No.: HY-118314
CAS No.: 156672-01-4
Synonyms: PD 144598
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CI-1015 is a potent CCK-B receptor antagonist.
Cat. No.: HY-B0477AS1
CAS No.: 1356020-03-5
Synonyms: CI-906-d5 hydrochloride
Cat. No.: HY-105235A
CAS No.: 124439-07-2
Synonyms: CI-977 hydrochloride
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Enadoline (CI-977) hydrochloride is a highly selective, brain-penetrating, and nonpeptide kappa-opioid receptor (KOR) agonist (Ki=1.25 nM). Antinociceptive effects .
Cat. No.: HY-139801
CAS No.: 80828-32-6
Synonyms: CI-907 hydrochloride
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Indolapril hydrochloride (CI-907) is an orally active nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor. Indolapril hydrochloride is highly specific in suppressing the contractile or pressor responses to Angiotensin I. Indolapril hydrochloride is a potent antihypertensive agent .
Cat. No.: HY-106305
CAS No.: 113457-05-9
Synonyms: CI 958
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Ledoxantrone (CI 958) is a DNA helicases inhibitor with an IC50 of 0.17 μM. Ledoxantrone can be used in the study of prostate cancer .
Cat. No.: HY-106305A
CAS No.: 119221-49-7
Synonyms: CI 958 trihydrochloride
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Ledoxantrone (CI 958) trihydrochloride is a DNA helicases inhibitor with an IC50 of 0.17 μM. Ledoxantrone trihydrochloride can be used in the study of prostate cancer .
Cat. No.: HY-106090A
CAS No.: 132937-88-3
Synonyms: CI-937 hydrochloride hydrate; DUP 937 hydrochloride hydrate
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Teloxantrone (CI-937; DUP 937) hydrochloride hydrate is a potent anticancer agent. Teloxantrone hydrochloride hydrate also is a DNA synthesis inhibitor .
Cat. No.: HY-B0477R
CAS No.: 82586-55-8
Synonyms: CI-906 (Standard)
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Quinapril (hydrochloride) (Standard) is the analytical standard of Quinapril (hydrochloride). This product is intended for research and analytical applications. Quinapril (hydrochloride) (CI-906) is a proagent that belongs to the angiotensin-converting enzyme (ACE) inhibitor class of medications.
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
