2 Results for "

MT7117

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "MT7117" in MCE Product Catalog:

Cat. No.: HY-109114
CAS No.: 1835256-48-8
Purity:  98.66%
Synonyms: MT-7117
Target:  

Melanocortin Receptor

Research Areas:  

Metabolic Disease

Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values of 8.16, 3.91, 1.14 and 0.251 nM for human (h), cynomolgus monkey (cm), mouse (m) and rat (r) MC1R, respectively. Dersimelagon shows good affinity for hMC1R and hMC4R with Ki values of 2.26, 32.9 nM, respectively. Dersimelagon can be used for the research of skin pigmentation .
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Cat. No.: HY-109114A
CAS No.: 2490660-87-0
Synonyms: MT-7117 phosphate
Target:  

Melanocortin Receptor

Research Areas:  

Metabolic Disease

Dersimelagon phosphate is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values of 8.16, 3.91, 1.14 and 0.251 nM for human (h), cynomolgus monkey (cm), mouse (m) and rat (r) MC1R, respectively. Dersimelagon phosphate shows good affinity for hMC1R and hMC4R with Ki values of 2.26, 32.9 nM, respectively. Dersimelagon phosphate can be used for the research of skin pigmentation .
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