22 Results for "

non-depolarizing

" in MedChemExpress (MCE) Product Catalog:
Products (22)

22 Results for "non-depolarizing" in MCE Product Catalog:

2
2 Cited Publications
Cat. No.: HY-17440
CAS No.: 119302-91-9
Synonyms: ORG 9426 Bromide
Target:  

nAChR

Rocuronium Bromide (ORG 9426 Bromide) is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia, to facilitate endotracheal intubation and to provide skeletal musclerelaxation during surgery or mechanical ventilation.
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1
1 Cited Publications
Cat. No.: HY-13596
CAS No.: 96946-42-8
Purity:  ≥98.0%
Synonyms: 51W89 besylate; Cisatracurium besilate
Target:  

nAChR Autophagy

Research Areas:  

Neurological Disease Cancer

Cisatracurium besylate (51W89) is a nondepolarizing neuromuscular blocking agent, antagonizing the action of acetylcholine by inhibiting neuromuscular transmission.
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1
1 Cited Publications
Cat. No.: HY-B0292A
CAS No.: 64228-81-5
Synonyms: BW-33A
Target:  

nAChR

Atracurium (BW-33A) besylate is a potent, competitive and non-depolarizing neuromuscular blocking agent. Atracurium besylate also is an AChR receptor antagonist. Atracurium besylate induces bronchoconstriction and neuromuscular blockade. Atracurium besylate promotes astroglial differentiation .
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Cat. No.: HY-B0118A
CAS No.: 50700-72-6
Synonyms: ORG NC 45
Target:  

nAChR

Research Areas:  

Neurological Disease Cancer

Vecuronium (ORG NC 45) bromide is a non-depolarizing neuromuscular blocking agent that also acts as a nicotinic acetylcholine receptor (nAChR) inhibitor, a muscle relaxant, and can be used for pre-surgical anesthesia .
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Cat. No.: HY-B1700A
CAS No.: 106861-44-3
Target:  

nAChR

Research Areas:  

Neurological Disease

Mivacurium dichloride is a benzylisoquinoline derivative and is a short-acting non-depolarizing neuromuscular blocking agent and skeletal muscle relaxant. Mivacurium dichloride couples with the nAChR to reduce or inhibit the depolarizing effect of acetylcholine on the terminal disc of the muscle cell .
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Cat. No.: HY-B0743A
CAS No.: 52212-02-9
Target:  

nAChR

Research Areas:  

Neurological Disease

Pipecuronium bromide is a potent long-acting nondepolarizing steroidal neuromuscular blocking agent (NMBA), and a bisquaternary ammonium compound. Pipecuronium bromide is a powerful competitive nAChR antagonist with a Kd of 3.06 μM .
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Cat. No.: HY-17033
CAS No.: 143558-00-3
Synonyms: Org-9426
Target:  

nAChR

Research Areas:  

Neurological Disease Cancer

Rocuronium (Org-9426) is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia.
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Cat. No.: HY-16423
CAS No.: 156137-99-4
Synonyms: Org 9487
Target:  

mAChR

Research Areas:  

Neurological Disease

Rapacuronium bromide (Org 9487), a non-depolarizing neuromuscular blocker, is an allosteric modulator of muscarinic acetylcholine receptor (mAChR) .
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Cat. No.: HY-A0258A
CAS No.: 7601-55-0
Synonyms: Metocurine iodide; Dimethylchondrocurarine iodide
Target:  

nAChR

Research Areas:  

Neurological Disease

Metubine (Metocurine iodide) is a non-depolarizing muscle relaxant. Metubine has neuromuscular blocking activities .
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Cat. No.: HY-125463
CAS No.: 142021-80-5
Target:  

nAChR

Research Areas:  

Neurological Disease

ANQ9040 is a steroidal relaxant. ANQ9040 is a relatively low-affinity and non-depolarizing nicotinic antagonist .
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Cat. No.: HY-B1700AR
CAS No.: 106861-44-3
Research Areas:  

Neurological Disease

Mivacurium (dichloride) (Standard) is the analytical standard of Mivacurium (dichloride). This product is intended for research and analytical applications. Mivacurium dichloride is a benzylisoquinoline derivative and is a short-acting non-depolarizing neuromuscular blocking agent and skeletal muscle relaxant. Mivacurium dichloride couples with the nAChR to reduce or inhibit the depolarizing effect of acetylcholine on the terminal disc of the muscle cell .
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Cat. No.: HY-A0215
CAS No.: 106819-53-8
Synonyms: BW-A 938U; Nuromax
Target:  

nAChR

Research Areas:  

Neurological Disease

Doxacurium chloride (BW A938U) is a potent non-depolarizing neuromuscular blocking agent. Doxacurium chloride binds to cholinergic receptors to antagonize acetylcholine, resulting in a block of neuromuscular transmission. Doxacurium chloride can be used for the research of neurological diseases .
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Cat. No.: HY-B0292
CAS No.: 64228-79-1
Synonyms: BW-33A free acid
tracurium (BW-33A free acid) is a potent, competitive and non-depolarizing neuromuscular blocking agent.Atracurium also is an AChR receptor antagonist. Atracurium induces bronchoconstriction and neuromuscular blockade. Atracurium promotes astroglial differentiation .
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Cat. No.: HY-17440R
CAS No.: 119302-91-9
Synonyms: ORG 9426 Bromide (Standard)
Research Areas:  

Neurological Disease Cancer

Rocuronium (Bromide) (Standard) is the analytical standard of Rocuronium (Bromide). This product is intended for research and analytical applications. Rocuronium Bromide (ORG 9426 Bromide) is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia, to facilitate endotracheal intubation and to provide skeletal musclerelaxation during surgery or mechanical ventilation.
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Cat. No.: HY-B0118AR
CAS No.: 50700-72-6
Synonyms: ORG NC 45 (Standard)
Research Areas:  

Neurological Disease Cancer

Vecuronium (bromide) (Standard) is the analytical standard of Vecuronium (bromide). This product is intended for research and analytical applications. Vecuronium (ORG NC 45) bromide is a non-depolarizing neuromuscular blocking agent that also acts as a nicotinic acetylcholine receptor (nAChR) inhibitor, a muscle relaxant, and can be used for pre-surgical anesthesia .
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Cat. No.: HY-B0292AR
CAS No.: 64228-81-5
Synonyms: BW-33A (Standard)
Atracurium (besylate) (Standard) is the analytical standard of Atracurium (besylate). This product is intended for research and analytical applications. Atracurium (BW-33A) besylate is a potent, competitive and non-depolarizing neuromuscular blocking agent. Atracurium besylate also is an AChR receptor antagonist. Atracurium besylate induces bronchoconstriction and neuromuscular blockade. Atracurium besylate promotes astroglial differentiation .
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Cat. No.: HY-13709
CAS No.: 213998-46-0
Synonyms: AV 4430A; GW 280430A
Research Areas:  

Neurological Disease

Gantacurium is an ultrashort-acting, nondepolarizing neuromuscular blocking agent that is degraded by nonenzymatic binding to L-cysteine under physiological conditions. Gantacurium causes a decrease in mean arterial pressure and an increase in heart rate .
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Cat. No.: HY-13596R
CAS No.: 96946-42-8
Synonyms: 51W89 besylate (Standard); Cisatracurium besilate (Standard)
Cisatracurium (besylate) (Standard) is the analytical standard of Cisatracurium (besylate). This product is intended for research and analytical applications. Cisatracurium besylate (51W89) is a nondepolarizing neuromuscular blocking agent, antagonizing the action of acetylcholine by inhibiting neuromuscular transmission.
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Cat. No.: HY-126175
CAS No.: 1212-37-9
Target:  

Endogenous Metabolite

Research Areas:  

Neurological Disease

Neostigmine iodide is a reversible acetylcholinesterase inhibitor with muscle tone-enhancing activity. Neostigmine iodide is primarily used to improve muscle function in patients with myasthenia gravis. Neostigmine iodide is also used in routine anesthesia to reverse the effects of nondepolarizing muscle relaxants such as rocuronium .
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Cat. No.: HY-182537
CAS No.: 119302-18-0
Target:  

Drug Derivative

Research Areas:  

Neurological Disease

Org 9616 bromide is a non-depolarizing neuromuscular blocker with a structure similar to Pancuroniam. Org 9616 bromide induces rapid-onset, short-duration neuromuscular blockade .
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