TS-021 free base
Based on 1 Customer Validation
DPP-IV-IN-1 is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV), a highly specific serine protease, with an IC50 of 4.6 nM.
Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.
- Pureté : 98.84%
- CAS No.: 625110-37-4
- Formule: C11H18FN3O2
- Masse moléculaire:243.28
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Stockage:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Activité biologique
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Chemical Information
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Solvant et solubilité
- Pureté et documentation
- Références
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Help & FAQs
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Activité biologique
Description
IC50 & Target
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DPP-4 |
In Vivo
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 625110-37-4
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Appearance Solid
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Masse moléculaire 243.28
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Formule C11H18FN3O2
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Color White to off-white
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SMILES
N#C[C@H]1N(C(CNC(C)(C)CO)=O)C[C@@H](F)C1
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Synonyms
DPP-IV-IN-1
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Solvant et solubilité
In Vitro:
DMSO : 200 mg/mL (822.09 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:
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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Working solution concentration: 0.22 mg/mL
Pureté et documentation
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Fiche technique (270 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Instruction de manipulation (2659 KB)
Références
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
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| DMSO | 1 mM | 4.1105 mL | 20.5523 mL | 41.1046 mL | 102.7614 mL |
| 5 mM | 0.8221 mL | 4.1105 mL | 8.2209 mL | 20.5523 mL | |
| 10 mM | 0.4110 mL | 2.0552 mL | 4.1105 mL | 10.2761 mL | |
| 15 mM | 0.2740 mL | 1.3702 mL | 2.7403 mL | 6.8508 mL | |
| 20 mM | 0.2055 mL | 1.0276 mL | 2.0552 mL | 5.1381 mL | |
| 25 mM | 0.1644 mL | 0.8221 mL | 1.6442 mL | 4.1105 mL | |
| 30 mM | 0.1370 mL | 0.6851 mL | 1.3702 mL | 3.4254 mL | |
| 40 mM | 0.1028 mL | 0.5138 mL | 1.0276 mL | 2.5690 mL | |
| 50 mM | 0.0822 mL | 0.4110 mL | 0.8221 mL | 2.0552 mL | |
| 60 mM | 0.0685 mL | 0.3425 mL | 0.6851 mL | 1.7127 mL | |
| 80 mM | 0.0514 mL | 0.2569 mL | 0.5138 mL | 1.2845 mL | |
| 100 mM | 0.0411 mL | 0.2055 mL | 0.4110 mL | 1.0276 mL |
TS-021 free base Related Classifications
HY-U00346 Related Classifications
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