Vestipitant mesylate
Vestipitant (GW597599) mesylate is a selective, orally active, and blood-brain barrier penetrant NK1 receptor antagonist. Vestipitant mesylate exhibits high affinity for the human NK1 receptor (pKi: 9.65). Vestipitant mesylate can be used in the research of diseases such as depression, anxiety disorders, and nausea and vomiting.
For research use only. We do not sell to patients.
- CAS No.: 334476-64-1
- Formula: C24H28F7N3O4S
- Molecular Weight:587.55
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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human NK1 9.65 (pKi) |
| NCT Number | Sponsor | Condition | Start Date |
Phase
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|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 334476-64-1
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Molecular Weight 587.55
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Formula C24H28F7N3O4S
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SMILES
O=C(N1CCNC[C@@H]1C2=CC=C(F)C=C2C)N([C@@H](C3=CC(C(F)(F)F)=CC(C(F)(F)F)=C3)C)C.CS(=O)(O)=O
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Synonyms
GW597599 mesylate; GW597599B
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Vestipitant mesylate Related Classifications
HY-12141 Related Classifications
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