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Cat. No.: HY-116484

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Way 100252

Way 100252 is a presynaptic GABA autoreceptor agonist. Way 100252 exerts its effect by inhibiting GABA release, and it suppresses GABA release induced by K⁺, Ca²⁺, Ouabain (HY-B1457) and electrical stimulation, with a more potent inhibitory effect on electrically evoked release. Way 100252 is used for studies related to GABAergic neurotransmission.

연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.

CAS No.: 129041-16-3
화학식: C₂₆H₂₅NO₂
분자량:383.48

보관:

Please store the product under the recommended conditions in the Certificate of Analysis.

Way 100252 Chemical Structure

CAS No.: 129041-16-3

Amount: USD 0.00

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- 제품 설명
- In Vitro
Chemical Information
순도&문서
References
Calculators
Help & FAQs
Classifications
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Biological Activity

제품 설명

In Vitro

Way 100252 dose-dependently inhibits the release of [³H] GABA evoked by various stimuli in cross-cut rat cerebral cortical slices, with pD₂ values of 5.8 (Ca²⁺), 7.4 (K⁺), 6.3 (electrical stimulation) and 6.0 (Ouabain (HY-B1457)) for different stimuli, respectively, and the maximum inhibitory effect ranges from 40% to 90%^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Related Protocols :

Ca²⁺ Staining Technique

Chemical Information

CAS No. 129041-16-3
분자량 383.48
화학식 C₂₆H₂₅NO₂
SMILES

O=C(CCCN(CC1=C2C=CC=CC2=CC=C1)CC3=C4C=CC=CC4=CC=C3)O
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.

순도&문서

Handling Instructions (2659 KB)

References

[1]. Dunlop J, et al. WAY 100252 inhibits evoked [3H]GABA release when tested against a number of release-inducing stimuli. Biochem Soc Trans. 1993 May;21(2):112S.

Calculators

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

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Molecular Weight Molecular Weight

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Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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MOQ

Minimum order quantity

100 mg

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