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  3. Nomegestrol

Nomegestrol 

Cat. No.: HY-105634
Handling Instructions

Nomegestrol is a potent and orally available progestin, acts as a selective full progesterone receptor agonist, with a Kd of 5.44 nM for rat uterine progesterone receptor, and has moderate antiandrogenic activity and strong antiestrogenic activity.

For research use only. We do not sell to patients.

Nomegestrol Chemical Structure

Nomegestrol Chemical Structure

CAS No. : 58691-88-6

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Description

Nomegestrol is a potent and orally available progestin, acts as a selective full progesterone receptor agonist, with a Kd of 5.44 nM for rat uterine progesterone receptor, and has moderate antiandrogenic activity and strong antiestrogenic activity.

IC50 & Target

Kd: 5.44 nM (Rat uterine progesterone receptor)[1]

In Vitro

Nomegestrol is a progestin, has high binding affinity at progesterone receptor, with a Kd of 5.44 nM for rat uterine progesterone receptor[1]. Nomegestrol acetate (NOMAC) is a higly selective progesterone receptor full agonist, but shows no or little binding affinity at other steroid receptors, such as the androgen and glucocorticoid receptors. Nomegestrol acetate has moderate antiandrogenic activity and strong antiestrogenic activity[2].

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
Molecular Weight

328.45

Formula

C₂₁H₂₈O₃

CAS No.

58691-88-6

SMILES

C[[email protected]@]12[[email protected]](CC[[email protected]]2(O)C(C)=O)([H])[[email protected]@]3([H])[[email protected]]([[email protected]]4([H])C(C(C)=C3)=CC(CC4)=O)([H])CC1

Shipping

Room temperature in continental US; may vary elsewhere

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This equation is commonly abbreviated as: C1V1 = C2V2

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× = ×
C1   V1   C2   V2

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Product Name:
Nomegestrol
Cat. No.:
HY-105634
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Nomegestrol

Cat. No.: HY-105634