1. PROTAC
  2. Ligand for Target Protein for PROTAC
  3. PROTAC Sirt2-binding moiety 1

PROTAC Sirt2-binding moiety 1 

Cat. No.: HY-107453
Handling Instructions

PROTAC Sirt2-binding moiety 1 is a selective and highly potent Sirtuin 2 (Sirt2) inhibitor, with an IC50 of 2.4 μM. For the development of sirtuin rearranging ligands (SirReals)-based PROTAC.

For research use only. We do not sell to patients.

PROTAC Sirt2-binding moiety 1 Chemical Structure

PROTAC Sirt2-binding moiety 1 Chemical Structure

CAS No. : 1862237-99-7

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 605 In-stock
Estimated Time of Arrival: December 31
5 mg USD 550 In-stock
Estimated Time of Arrival: December 31
10 mg USD 850 In-stock
Estimated Time of Arrival: December 31
50 mg USD 2650 In-stock
Estimated Time of Arrival: December 31
100 mg USD 3650 In-stock
Estimated Time of Arrival: December 31
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Description

PROTAC Sirt2-binding moiety 1 is a selective and highly potent Sirtuin 2 (Sirt2) inhibitor, with an IC50 of 2.4 μM. For the development of sirtuin rearranging ligands (SirReals)-based PROTAC[1].

IC50 & Target

IC50: 2.4 μM (Sirt2)[1].

Molecular Weight

424.54

Formula

C₂₁H₂₀N₄O₂S₂

CAS No.

1862237-99-7

SMILES

O=C(NC1=NC=C(CC2=CC=CC(OCC#C)=C2)S1)CSC3=NC(C)=CC(C)=N3

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Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Product Name:
PROTAC Sirt2-binding moiety 1
Cat. No.:
HY-107453
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