1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. Adrenergic Receptor
  4. β adrenergic receptor Isoform
  5. β adrenergic receptor Antagonist

β adrenergic receptor Antagonist

β adrenergic receptor Antagonists (27):

Cat. No. Product Name Effect Purity
  • HY-B0573
    Propranolol hydrochloride
    Antagonist 99.97%
    Propranolol hydrochloride is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively.
  • HY-105124
    Bufuralol
    Antagonist 98.26%
    Bufuralol (Ro 3-4787) is a potent non-selective, orally active β-adrenoreceptor antagonist with partial agonist activity.
  • HY-P3557
    Mibenratide
    Antagonist
    Mibenratide, a small cyclic peptide, is an adrenergic β1 receptor antagonist.
  • HY-17503C
    Metoprolol fumarate
    Antagonist
    Metoprolol fumarate (CGP 2175C) is an orally active, selective β1-adrenoceptor antagonist.
  • HY-17498
    Atenolol
    Antagonist 99.82%
    Atenolol ((RS)-Atenolol) is a cardioselective β1-adrenergic receptor blocker, with a Ki of 697 nM atβ1-adrenoceptor in guine pig left ventricle membrane.
  • HY-B0573B
    Propranolol
    Antagonist 99.87%
    Propranolol is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively.
  • HY-17503
    Metoprolol
    Antagonist 99.89%
    Metoprolol is an orally active, selective β1-adrenoceptor antagonist.
  • HY-17503A
    Metoprolol succinate
    Antagonist 99.90%
    Metoprolol succinate is an orally active, selective β1-adrenoceptor antagonist.
  • HY-17497A
    Acebutolol hydrochloride
    Antagonist 99.97%
    Acebutolol hydrochloride is an orally active β1 adrenergic receptor (β1AR) antagonist.
  • HY-121383
    Labetalol
    Antagonist 99.88%
    Labetalol (AH5158) is an orally active selective α1- and non-selective β-adrenergic receptors competitive antagonist.
  • HY-105124A
    Bufuralol hydrochloride
    Antagonist ≥99.0%
    Bufuralol (Ro 3-4787) hydrochloride is a potent non-selective, orally active β-adrenoreceptor antagonist with partial agonist activity.
  • HY-B1486
    Oxprenolol hydrochloride
    Antagonist 99.86%
    Oxprenolol hydrochloride (Ba 39089) is an orally bioavailable β-adrenergic receptor (β-AR) antagonist with a Ki of 7.10 nM in a radioligand binding assay using rat heart muscle.
  • HY-B1035
    Levobunolol hydrochloride
    Antagonist 99.75%
    Levobunolol (l-Bunolol) hydrochloride is a potent and nonselective β-adrenergic receptor antagonist.
  • HY-121567
    Metipranolol
    Antagonist 98.36%
    Metipranolol is a nonselective and orally active β-adrenergic receptor antagonist.
  • HY-107327
    Carazolol
    Antagonist ≥99.0%
    Carazolol is a β12 adrenoceptor antagonist of high potency used in the research of hypertension.
  • HY-17503B
    Metoprolol tartrate
    Antagonist
    Metoprolol tartrate is an orally active, selective β1-adrenoceptor antagonist.
  • HY-B1562C
    Bopindolol fumarate
    Antagonist
    Bopindolol ((±)-Bopindolol) fumarate is an orally active antagonist of β-adrenoceptors (ARs) with partial agonist activity.
  • HY-119873
    Celiprolol
    Antagonist
    Celiprolol (REV 5320) is a potent, cardioselective and orally active β1-andrenoceptor r antagonist with partial β2 agonist activity, with Ki values of 0.14-8.3 μM.
  • HY-B1486A
    Oxprenolol
    Antagonist
    Oxprenolol (Ba 39089 free base) is an orally bioavailable β-adrenergic receptor (β-AR) antagonist with a Ki of 7.10 nM in a radioligand binding assay using rat heart muscle.
  • HY-B1562
    Bopindolol
    Antagonist
    Bopindolol ((±)-Bopindolol) is an orally active antagonist of β-adrenoceptors (ARs) with partial agonist activity.