Drug Metabolite
Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.
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Drug Metabolite Related Products (2022)
Related Products (2022)
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Antibodies (1)
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Related Compound Screening Libraries (1)
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Mephedrone metabolite hydrochloride ((±)-ephedrine stereochemistry)
0 ImagesCat. No.: HY-W035375CAS No.: 117342-78-6Mephedrone metabolite hydrochloride ((±)-ephedrine stereochemistry) is a metabolite of Mephedrone.
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4-Hydroxyalprenolol
0 ImagesCat. No.: HY-177977CAS No.: 54175-82-5Synonyms: Alp2b4-Hydroxyalprenolol (Alp2b) is a metabolite of β-receptor blocker Alprenolol (HY-B1517).
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Para-hydroxy 2-methyl AP-237 hydrochloride
0 ImagesCat. No.: HY-175054CAS No.: 2981814-36-0Synonyms: 4'-Hydroxy 2-methyl AP-237 hydrochloride; p-Hydroxy 2-methyl AP-237 hydrochloridePara-hydroxy 2-methyl AP-237 (4'-Hydroxy 2-methyl AP-237, p-Hydroxy 2-methyl AP-237) hydrochloride is a metabolite of 2-methyl AP-237.
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6-O-Desmethyl donepezil-d7
0 ImagesCat. No.: HY-133925S2CAS No.: 1261396-76-2Synonyms: 6-o-Desmethyldonepezil-d76-O-Desmethyl donepezil-d7 is deuterated labeled 6-O-Desmethyl donepezil.
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CNDAC
0 ImagesCat. No.: HY-16445ACAS No.: 135598-68-4CNDAC is a metabolite of the orally active agent Sapacitabine (HY-16445), and a nucleoside analog. CNDAC induces DNA damage and apoptosis.
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Modafinil acid (Standard)
0 ImagesSynonyms: CRL-40467 (Standard)Modafinil acid (Standard) (CRL-40467 (Standard)) is the analytical standard of Modafinil acid (HY-W103882). This product is intended for research and analytical applications. Modafinil acid is the metabolite of Modafinil.
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Captopril EP Impurity E
0 ImagesCat. No.: HY-137772CAS No.: 23500-15-4Captopril EP Impurity E is an impurity of Captopril. Captopril (SQ-14534), antihypertensive agent, is a thiol-containing competitive, orally active angiotensin-converting enzyme (ACE) inhibitor (IC50=0.025 μM).
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4-Hydroxyphenylbutazone (Standard)
0 ImagesCat. No.: HY-139199RCAS No.: 16860-43-84-Hydroxyphenylbutazone (Standard) is the analytical standard of 4-Hydroxyphenylbutazone. This product is intended for research and analytical applications. 4-Hydroxyphenylbutazone is a metabolite of Phenylbutazone. Phenylbutazone, a nonsteroidal anti-inflammatory agent (NSAID), is an efficient reducing cofactor for the peroxidase activity of prostaglandin H synthase (PHS).
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Dimethyl sulfone (Standard)
0 ImagesDimethyl sulfone (Standard) is the analytical standard of Dimethyl sulfone. This product is intended for research and analytical applications. Dimethyl sulfone (Methyl Sulfonyl Methane) is a metabolic product of endogenous methanethiol metabolism and intestinal bacterial metabolism. Dimethyl sulfone inhibits choriocapillary endothelial (CCE) cell proliferation, also has many biological effects, including antiinflammatory, antioxidant, and local anesthetic effects that could be neuroprotective.
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7-Aminoflunitrazepam-d7
0 ImagesCat. No.: HY-116687S7-Aminoflunitrazepam-d7 is deuterium labeled 7-Aminoflunitrazepam.
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Monobutyl phosphate-d9
0 ImagesCat. No.: HY-W704657CAS No.: 156213-20-6Monobutyl phosphate-d9 is the deuterium labeled Monobutyl phosphate (HY-N7143). Monobutyl phthalate, a major metabolite of dibutyl phthalate (DBP), possesses antiandrogenic effects.
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Cefdaloxime
0 ImagesCat. No.: HY-W744633CAS No.: 80195-36-4Cefdaloxime is an orally active cephalosporin and HR-916 ester metabolite. Cefdaloxime has a broad spectrum of activity against pathogens such as the majority of members of the family Enterobacteriaceae, staphylococci, Streptococcus spp., Neisseria gonorrhoeae, Moraxella catarrhalis, Haemophilus influenzae.
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6-Hydroxy Chlorzoxazone-d2
0 ImagesCat. No.: HY-W016221SCAS No.: 1432065-00-36-Hydroxy Chlorzoxazone-d2 is deuterium labeled 6-Hydroxy Chlorzoxazone. 6-Hydroxy Chlorzoxazone is a metabolite of Chlorzoxazone (HY-B1462). Chlorzoxazone is a centrally acting muscle relaxant used to treat muscle spasm and the resulting pain or discomfort.
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3-Methylcrotonyl CoA
0 Images3-Methylcrotonyl CoA is a key metabolic intermediate in the leucine degradation pathway, converted to 3-Methylglutaconyl CoA by 3-Methylcrotonyl CoA Carboxylase. Normally, 3-Methylglutaconyl CoA is catalyzed by 3-Methylglutaconyl-CoA Hydratase into 3-Hydroxy-3-methylglutaryl-CoA (HMG CoA). However, mutations in 3-Methylglutaconyl-CoA Hydratase lead to the accumulation of 3-Methylglutaconyl CoA, causing metabolic disorders associated with 3MGA-uria. 3-Methylcrotonyl CoA is useful for research into metabolic diseases related to the leucine degradation pathway.
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Acetaminophen glucuronide (Standard)
0 ImagesCat. No.: HY-113083RCAS No.: 16110-10-4Synonyms: APAP-glu (Standard)Acetaminophen glucuronide (Standard) is the analytical standard of Acetaminophen glucuronide. This product is intended for research and analytical applications. Acetaminophen glucuronide (APAP-glu) is an inactive glucuronide metabolite of Acetaminophen (HY-66005). Acetaminophen is a selective cyclooxygenase-2 (COX-2) inhibitor and a potent hepatic N-acetyltransferase 2 (NAT2) inhibitor.
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4-Methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-5-carboxylic acid
![4-Methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-5-carboxylic acid](https://file.medchemexpress.com/product_pic/hy-w158239.gif "Click to View 4-Methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-5-carboxylic acid Product Detail")
0 ImagesCat. No.: HY-W158239CAS No.: 144059-86-9
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Mycophenolic acid acyl-β-D-glucuronide
0 ImagesCat. No.: HY-W587775CAS No.: 99043-04-6Synonyms: Acyl-MPAGMycophenolic acid acyl-β-D-glucuronide (Acyl-MPAG) is a metabolite of Mycophenolic acid (MPA) , an immunosuppressant.
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Ribavirin carboxylic acid (Standard)
0 ImagesCat. No.: HY-145991RCAS No.: 39925-19-4
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Teriflunomide (Standard)
0 ImagesSynonyms: A77 1726 (Standard)Teriflunomide (Standard) is the analytical standard of Teriflunomide. This product is intended for research and analytical applications. Teriflunomide is the active metabolite of leflunomide, an approved therapy for rheumatoid arthritis. It inhibits pyrimidine synthesis and therefore potently decreases T cell and B cell proliferation.
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PD 109488 (Standard)
0 ImagesCat. No.: HY-114547RCAS No.: 103733-49-9Synonyms: Quinapril Diketopiperazine (Standard)PD 109488 (Standard) is the analytical standard of PD 109488. This product is intended for research and analytical applications. PD 109488 is a quinapril diketopiperazine metabolite.
