1. Signaling Pathways
  2. Vitamin D Related/Nuclear Receptor
  3. Estrogen Receptor/ERR
  4. Estrogen receptor Isoform
  5. Estrogen receptor Modulator

Estrogen receptor Modulator

Estrogen receptor Modulators (8):

Cat. No. Product Name Effect Purity
  • HY-13757A
    Tamoxifen
    Modulator 99.92%
    Tamoxifen (ICI 47699) is an orally active, selective estrogen receptor modulator (SERM) which blocks estrogen action in breast cells and can activate estrogen activity in other cells, such as bone, liver, and uterine cells.
  • HY-16950
    4-Hydroxytamoxifen
    Modulator 99.96%
    4-Hydroxytamoxifen ((Z)-4-Hydroxytamoxifen) is an orally active, selective estrogen receptor modulator (SERM).
  • HY-13757
    Tamoxifen Citrate
    Modulator 99.95%
    Tamoxifen Citrate (ICI 46474) is an orally active, selective estrogen receptor modulator (SERM) which blocks estrogen action in breast cells and can activate estrogen activity in other cells, such as bone, liver, and uterine cells.
  • HY-16950A
    (E/Z)-4-Hydroxytamoxifen
    Modulator 99.60%
    (E/Z)-4-Hydroxytamoxifen (Afimoxifene) is a racemic compound of (Z)-4-Hydroxytamoxifen and (E)-4-Hydroxytamoxifen isomers.
  • HY-13757AS
    Tamoxifen-d5
    Modulator 99.99%
    Tamoxifen-d5 (ICI 47699-d5) is a deuterium labeled Tamoxifen.
  • HY-16950B
    (E)-4-Hydroxytamoxifen
    Modulator 98.27%
    (E)-4-Hydroxytamoxifen ((E)-Afimoxifene), the less active isomer of (Z)-4-hydroxytamoxifen, is an estrogen receptor modulator.
  • HY-13738
    Raloxifene
    Modulator
    Raloxifene (Keoxifene) is a benzothiophene-derived selective estrogen receptor modulator (SERM).
  • HY-116896
    LY117018
    Modulator
    LY117018, a Raloxifene analog, is a selective estrogen receptor modulator.