1. Signaling Pathways
  2. Cell Cycle/DNA Damage
    Epigenetics
  3. HDAC
  4. HDAC Isoform
  5. HDAC Antagonist

HDAC Antagonist

HDAC Antagonists (2):

Cat. No. Product Name Effect Purity
  • HY-131961
    Triciferol
    Antagonist 98.61%
    Triciferol functions as a multiple ligand with combined VDR agonist and HDAC antagonist activities. Triciferol binds directly to the VDR (IC50=87 nM), and functions as an agonist with 1,25D-like potency on several 1,25D target genes. Triciferol induces marked tubulin hyperacetylation, and augments histone acetylation. Antiproliferative and cytotoxic activities.
  • HY-155697
    SGC-UBD253
    Antagonist
    SGC-UBD253 is a potent HDAC6-UBD antagonist. SGC-UBD253 can be used in research of cancer.