Vasopressin Receptor Antagonist
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Atosiban
0 ImagesSynonyms: RW22164; RWJ22164Atosiban (RW22164; RWJ22164) is a nonapeptide competitive vasopressin/oxytocin receptor antagonist, and is a desamino-oxytocin analogue. Atosiban is the main tocolytic agent and has the potential for spontaneous preterm labor research.
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Atosiban acetate
0 ImagesSynonyms: RW22164 acetate; RWJ22164 acetateAtosiban acetate (RW22164 acetate;RWJ22164 acetate) is a nonapeptide competitive vasopressin/oxytocin receptor antagonist, and is a desamino-oxytocin analogue. Atosiban is the main tocolytic agent and has the potential for spontaneous preterm labor research.
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Nelivaptan
0 ImagesSynonyms: SSR-149415Nelivaptan (SSR-149415) is a selective and orally active vasopressin V1b receptor antagonist (Ki: 3.7 and 1.3 nM for native and recombinant rat V1b receptors, respectively). Nelivaptan inhibits arginine vasopressin (AVP)-induced Ca2+ increase and corticotropin secretion. Nelivaptan can be used for research of stress, anxiety and depression.
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Atosiban acetate solution
0 ImagesCat. No.: HY-FL17572ACAS No.: 914453-95-5Synonyms: RW22164 acetate solution; RWJ22164 acetate solutionAtosiban acetate solution is mainly composed of Atosiban acetate (HY-17572A). Atosiban acetate (RW22164 acetate;RWJ22164 acetate) is a nonapeptide competitive vasopressin/oxytocin receptor antagonist, and is a desamino-oxytocin analogue. Atosiban is the main tocolytic agent and has the potential for spontaneous preterm labor research.
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Atosiban-d5 TFA
0 ImagesCat. No.: HY-17572SSynonyms: RW22164-d5 TFA; RWJ22164-d5 TFAAtosiban-d5 TFA (RW22164-d5 TFA) is the deuterium labeled Atosiban TFA. Atosiban (RW22164; RWJ22164) is a nonapeptide competitive vasopressin/oxytocin receptor antagonist, and is a desamino-oxytocin analogue. Atosiban is the main tocolytic agent and has the potential for spontaneous preterm labor research.
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Fidinvaptan
0 ImagesCat. No.: HY-187869CAS No.: 2826938-65-0Fidinvaptan is a Vasopressin receptor antagonist.
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Vasopressin V2 receptor antagonist 2
0 ImagesVasopressin V2 receptor antagonist 2 (Compound 33) is an antagonist of the arginine vasopressin V2 receptor (V2R) with a Ki value of 6.2 nM. Vasopressin V2 receptor antagonist 2 can effectively reduce cAMP levels, thereby inhibiting the growth of renal cysts[1].
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Brezivaptan
0 ImagesCat. No.: HY-159507CAS No.: 1370444-22-6Synonyms: Brezivaptanum; TH1773; TS-121Brezivaptan (Brezivaptanum; TH1773; TS-121) is a vasopressin receptor antagonist.
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Tolvaptan phosphate ester sodium
0 ImagesTolvaptan phosphate ester sodium, a prodrug of Tolvaptan (HY-17000), can be used in the study of cardiac edema. Tolvaptan is a selective, competitive and orally active vasopressin receptor 2 (V2R) antagonist with an IC50 of 1.28 μM for the inhibition of arginine vasopressin (AVP)-induced platelet aggregation.
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JKC 301
0 ImagesCat. No.: HY-P4201CAS No.: 136553-96-3JKC 301 is a selective Endothelin A receptor antagonist. JKC 301 attenuates the pressor effects of nicotine in rats. JKC 301 can be used to study cardiovascular disease caused by smoking.
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Enuvaptan
0 ImagesCat. No.: HY-139572CAS No.: 2145062-48-0Synonyms: BAY-2327949Enuvaptan (BAY-2327949) is a vasopressin receptor antagonist and has the potential for research into renal and cardiovascular diseases.
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Dp[Tyr(methyl)2,Arg8]-Vasopressin
![Dp[Tyr(methyl)2,Arg8]-Vasopressin](https://file.medchemexpress.com/product_pic/hy-p3213.gif "Click to View Dp[Tyr(methyl)2,Arg8]-Vasopressin Product Detail")
0 ImagesCat. No.: HY-P3213CAS No.: 67269-08-3Dp[Tyr(methyl)2,Arg8]-Vasopressin is a non-selective peptide arginine vasopressin Vlb receptor antagonist.
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2-(3-Trifluoromethylphenyl)glycine hydrochloride
0 ImagesCat. No.: HY-W104304CAS No.: 1134915-25-52-(3-Trifluoromethylphenyl)glycine hydrochloride is a precursor of substituted 2-acetamido-5-aryl-l, 2,4-triazolones. Substituted 2-acetamido-5-aryl-l, 2,4-triazolones are dual V1a/V2 receptor antagonists and can be used in cardiovascular disease research.
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Satavaptan
0 ImagesCat. No.: HY-18344CAS No.: 185913-78-4Synonyms: SR 121463Satavaptan (SR 121463) is an antagonist for vasopressin V2 receptor. Satavaptan regulates the vasopressin regulated phosphopeptides and vasopressin-mediated signaling pathway. Satavaptan is potential in ameliorating hyponatremia.
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Tolmesoxide
0 ImagesCat. No.: HY-107037CAS No.: 38452-29-8Synonyms: RX71107Tolmesoxide (RX71107) is a peripheral vascular dilator with blood pressure lowering activity. Tolmesoxide has shown direct vasodilation in the human forearm arterial bed and dorsal hand vein. Tolmesoxide can dose-dependently increase blood flow in the forearm and produce dilation during contraction of the dorsal hand veins. Tolmesoxide can be used to study high blood pressure and angina.
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Ribuvaptan
0 ImagesCat. No.: HY-16783CAS No.: 1245620-47-6Ribuvaptan is a vasopressin receptor antagonist. Ribuvaptan can be used for the study of Heart failure.
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Elsovaptan
0 ImagesCat. No.: HY-172427CAS No.: 2296801-25-5Elsovaptan is the antagonist for vasopressin receptor that can be used in researchs of Alzheimer disease.
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