2. GPCR/G Protein
  3. Vasopressin Receptor
  4. Tolvaptan phosphate ester sodium

Tolvaptan phosphate ester sodium, a prodrug of Tolvaptan (HY-17000), can be used in the study of cardiac edema. Tolvaptan is a selective, competitive and orally active vasopressin receptor 2 (V2R) antagonist with an IC50 of 1.28 μM for the inhibition of arginine vasopressin (AVP)-induced platelet aggregation.

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Tolvaptan phosphate ester sodium Chemical Structure

Tolvaptan phosphate ester sodium Chemical Structure

CAS No. : 942619-79-6

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Tolvaptan phosphate ester sodium Related Antibodies

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Description

Tolvaptan phosphate ester sodium, a prodrug of Tolvaptan (HY-17000), can be used in the study of cardiac edema. Tolvaptan is a selective, competitive and orally active vasopressin receptor 2 (V2R) antagonist with an IC50 of 1.28 μM for the inhibition of arginine vasopressin (AVP)-induced platelet aggregation[1][2].

Molecular Weight

572.88

Formula

C26H24ClN2Na2O6P
CAS No.
SMILES

O=C(C1=C(C)C=CC=C1)NC2=CC=C(C(C)=C2)C(N3C4=CC=C(C=C4C(CCC3)OP(O[Na])(O[Na])=O)Cl)=O
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Room temperature in continental US; may vary elsewhere.
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Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Tolvaptan phosphate ester sodium Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Tolvaptan phosphate ester942619-79-6Vasopressin ReceptorAVPvasopressin receptorcardiac edemaInhibitorinhibitorinhibit

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