1. Membrane Transporter/Ion Channel
  2. Potassium Channel

VU0529331 

Cat. No.: HY-112705
Handling Instructions

VU0529331 is a modestly selective non-GIRK1-containing G protein-gated, inwardly-rectifying, potassium channel (non-GIRK1/X) activator, with EC50s of 5.1 µM and 5.2 µM for GIRK2 and GIRK1/2 in HEK293 cells, respectively, also effective on GIRK4 homomeric channel.

For research use only. We do not sell to patients.

VU0529331 Chemical Structure

VU0529331 Chemical Structure

CAS No. : 1286725-49-2

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  • Biological Activity

  • Technical Information

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  • References

Description

VU0529331 is a modestly selective non-GIRK1-containing G protein-gated, inwardly-rectifying, potassium channel (non-GIRK1/X) activator, with EC50s of 5.1 µM and 5.2 µM for GIRK2 and GIRK1/2 in HEK293 cells, respectively, also effective on GIRK4 homomeric channel[1].

IC50 & Target

EC50: 5.1 µM (GIRK2), 5.2 µM (GIRK1/2)[1]

References
Molecular Weight

384.43

Formula

C₂₂H₂₀N₆O

CAS No.

1286725-49-2

SMILES

O=C(C1=NC=CN=C1)N2CC3=C(N4C=CC=C4)N(C5=CC(C)=C(C)C=C5)N=C3C2

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
VU0529331
Cat. No.:
HY-112705
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VU0529331

Cat. No.: HY-112705