1. Membrane Transporter/Ion Channel
  2. Potassium Channel
  3. VU0529331

VU0529331 

Cat. No.: HY-112705 Purity: >99.0%
Handling Instructions

VU0529331 is a modestly selective non-GIRK1-containing G protein-gated, inwardly-rectifying, potassium channel (non-GIRK1/X) activator, with EC50s of 5.1 µM and 5.2 µM for GIRK2 and GIRK1/2 in HEK293 cells, respectively, also effective on GIRK4 homomeric channel.

For research use only. We do not sell to patients.

VU0529331 Chemical Structure

VU0529331 Chemical Structure

CAS No. : 1286725-49-2

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1 mg USD 180 In-stock
Estimated Time of Arrival: December 31
5 mg USD 540 Get quote
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Based on 1 publication(s) in Google Scholar

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Description

VU0529331 is a modestly selective non-GIRK1-containing G protein-gated, inwardly-rectifying, potassium channel (non-GIRK1/X) activator, with EC50s of 5.1 µM and 5.2 µM for GIRK2 and GIRK1/2 in HEK293 cells, respectively, also effective on GIRK4 homomeric channel[1].

IC50 & Target

EC50: 5.1 µM (GIRK2), 5.2 µM (GIRK1/2)[1]

Molecular Weight

384.43

Formula

C₂₂H₂₀N₆O

CAS No.

1286725-49-2

SMILES

O=C(C1=NC=CN=C1)N2CC3=C(N4C=CC=C4)N(C5=CC(C)=C(C)C=C5)N=C3C2

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
In solvent -80°C 6 months
  -20°C 1 month
References

Purity: >99.0%

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Keywords:

VU0529331VU 0529331VU-0529331Potassium ChannelKcsAInhibitorinhibitorinhibit

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