A2A/A3 AR antagonist-1
A2A/A3 AR antagonist-1 (compound 23) is a dual A2A/A3 adenosine receptor (AR) fluorescent ligand, with Kis of 90 nM and 31.8 nM for hA2A AR and hA3 AR, respectively.
For research use only. We do not sell to patients.
- CAS No.: 1448221-36-0
- Formula: C56H71N15O12S2
- Molecular Weight:1210.39
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All Adenosine Receptor Isoforms
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Biological Activity
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hA2AAR 90 nM (Ki) |
hA3 31.8 nM (Ki) |
Chemical Information
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CAS No. 1448221-36-0
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Molecular Weight 1210.39
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Formula C56H71N15O12S2
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SMILES
CN1C=C2C(N=C(N3N=C(N=C23)C4=CC=CO4)NC(CCCC5=CN(N=N5)CCCCCCNC(C6=CC(C([O-])=O)=C(C=C6)C7=C8C=CC(C(S(=O)([O-])=O)=C8OC9=C(C(N)=CC=C97)S(=O)([O-])=O)=[NH2+])=O)=O)=N1.CC[NH+](CC)CC.CC[NH+](CC)CC
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
A2A/A3 AR antagonist-1 Related Classifications
HY-147541 Related Classifications
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