1. GPCR/G Protein
  2. Adenosine Receptor
  3. A2A/A3 AR antagonist-1

A2A/A3 AR antagonist-1 

Cat. No.: HY-147541
Handling Instructions

A2A/A3 AR antagonist-1 (compound 23) is a dual A2A/A3 adenosine receptor (AR) fluorescent ligand, with Kis of 90 nM and 31.8 nM for hA2A AR and hA3 AR, respectively.

For research use only. We do not sell to patients.

A2A/A3 AR antagonist-1 Chemical Structure

A2A/A3 AR antagonist-1 Chemical Structure

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Description

A2A/A3 AR antagonist-1 (compound 23) is a dual A2A/A3 adenosine receptor (AR) fluorescent ligand, with Kis of 90 nM and 31.8 nM for hA2A AR and hA3 AR, respectively[1].

IC50 & Target[1]

hA2AAR

90 nM (Ki)

hA3

31.8 nM (Ki)

Molecular Weight

1210.39

Formula

C56H71N15O12S2

SMILES

CN1C=C2C(N=C(N3N=C(N=C23)C4=CC=CO4)NC(CCCC5=CN(N=N5)CCCCCCNC(C6=CC(C([O-])=O)=C(C=C6)C7=C8C=CC(C(S(=O)([O-])=O)=C8OC9=C(C(N)=CC=C97)S(=O)([O-])=O)=[NH2+])=O)=O)=N1.CC[NH+](CC)CC.CC[NH+](CC)CC

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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A2A/A3 AR antagonist-1
Cat. No.:
HY-147541
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