[Ala17]-MCH TFA
[Ala17]-MCH TFA, a MCH analogue (HY-P1525A), is a selective ligand for MCHR1 (Ki=0.16 nM) over MCHR2 (Ki=34 nM). [Eu3+ chelate-labeled [Ala17]-MCH shows high affnity for MCHR1 (Kd=0.37 nM) while has little demonstrable binding affnity for MCHR2.
For research use only. We do not sell to patients.
- Formula: C99H156F3N29O28S4
- Molecular Weight:2385.73
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Ki: 0.16 nM (MCHR1)Ki: 34 nM (MCHR2)[1]
Chemical Information
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Molecular Weight 2385.73
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Formula C99H156F3N29O28S4
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Sequence
Asp-Phe-Asp-Met-Leu-Arg-Cys-Met-Leu-Gly-Arg-Val-Tyr-Arg-Pro-Cys-Ala-Gln-Val (Disulfide bridge:Cys7-Cys16)
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Sequence Shortening
DFDMLRCMLGRVYRPCAQV (Disulfide bridge:Cys7-Cys16)
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)