VU6036864
VU6036864 (compound 45) is an orally active, selective mAChR M5 antagonist with IC50=20 nM for human M5. VU6036864 is >500-fold selective for human M1-4, with BBB characteristic and high oral bioavailability (%F>100%).
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- CAS. Nr.: 2746406-36-8
- Formel: C15H12D4ClN5O3S
- Molecular Weight:385.86
-
Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biologische Aktivität
IC50: 20 nM (human mAChR M5)[1]
1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.
Chemical Information
-
CAS. Nr. 2746406-36-8
-
Unlabeled Cas 2746405-41-2
-
Molecular Weight 385.86
-
Formel C15H12D4ClN5O3S
-
SMILES
CC1=NC=C(S(=O)(N2C([2H])([2H])CC(C3=CN4C(C=C3Cl)=NC=N4)CC2([2H])[2H])=O)O1
-
Versand
Room temperature in continental US; may vary elsewhere.
-
Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)