BNTX maleate
Based on 1 Customer Validation
BNTX (7-Benzylidenenaltrexone) maleate is a δ1-opioid receptor antagonist with the Kis of 0.1, 10.8, 13.3, and 58.6 nM for δ1, δ2-, μ-, and κ-opioid receptor, respectively. BNTX maleate shows antinociceptive activity.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度 : 98.2%
- CAS 番号: 864461-31-4
- 分子式: C31H31NO8
- 分子量:545.58
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保管条件:
-20°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
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HY-P0210
DAMGOμ-OPR Agonist -
![[Leu5]-Enkephalin](https://file.medchemexpress.com/product_pic/hy-p0288.gif)
HY-P0288
[Leu5]-EnkephalinEndogenous Metabolite -
HY-101202
SNC80δ-opioid Receptor Agonist -
HY-P1334
DPDPEDOR Agonist -
HY-105343
BW-180COpioid Receptor Agonist -
HY-P1333
Dynorphin AKOR Agonist -
HY-100903
Norbinaltorphimine dihydrochlorideκ-opioid receptor Antagonist -
HY-P1335
CTAPμ Opioid Receptor Antagonist -
HY-13243
Alvimopanμ-opioid Receptor Antagonist -
HY-13274
JTC-801Opioid Receptor Antagonist -
HY-13044
ADL-5859 hydrochlorideOpioid Receptor Agonist -
HY-101230
ICI 174864δ-opioid receptor Antagonist
Opioid Receptor アイソフォーム固有の製品をすべて表示
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生物活性
製品説明
化学情報
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CAS 番号 864461-31-4
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性状 Solid
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分子量 545.58
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分子式 C31H31NO8
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Color White to off-white
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SMILES
O[C@@]1(C/C2=C\C3=CC=CC=C3)[C@]4([C@@](C2=O)([H])OC5=C6O)C5=C(C=C6)C[C@@]1([H])N(CC7CC7)CC4.OC(/C=C\C(O)=O)=O
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別名
7-Benzylidenenaltrexone maleate
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
-20°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
純度とドキュメンテーション
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データシート (273 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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取扱説明書 (2659 KB)
参考文献
[1]. Portoghese PS, et al. A highly selective delta 1-opioid receptor antagonist: 7-benzylidenenaltrexone. Eur J Pharmacol. 1992;218(1):195-196. [Content Brief]
[2]. House RV, et al. Suppression of immune function by non-peptidic delta opioid receptor antagonists. Neurosci Lett. 1995 Sep 29;198(2):119-22. [Content Brief]
[3]. Miyata Y, et al. Opioid δ₁ receptor antagonist 7-benzylidenenaltrexone as an effective resistance reverser for chloroquine-resistant Plasmodium chabaudi. Bioorg Med Chem Lett. 2011 Aug 15;21(16):4710-2. [Content Brief]
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
BNTX maleate 関連分類
HY-101307 関連分類
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