BNTX maleate
Based on 1 Customer Validation
BNTX (7-Benzylidenenaltrexone) maleate is a δ1-opioid receptor antagonist with the Kis of 0.1, 10.8, 13.3, and 58.6 nM for δ1, δ2-, μ-, and κ-opioid receptor, respectively. BNTX maleate shows antinociceptive activity.
For research use only. We do not sell to patients.
- Purity: 98.2%
- CAS No.: 864461-31-4
- Formula: C31H31NO8
- Molecular Weight:545.58
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Storage:
-20°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All Opioid Receptor Isoforms
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Biological Activity
Chemical Information
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CAS No. 864461-31-4
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Appearance Solid
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Molecular Weight 545.58
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Formula C31H31NO8
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Color White to off-white
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SMILES
O[C@@]1(C/C2=C\C3=CC=CC=C3)[C@]4([C@@](C2=O)([H])OC5=C6O)C5=C(C=C6)C[C@@]1([H])N(CC7CC7)CC4.OC(/C=C\C(O)=O)=O
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Synonyms
7-Benzylidenenaltrexone maleate
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
-20°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
Purity & Documentation
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Data Sheet (273 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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Handling Instructions (2659 KB)
References
[1]. Portoghese PS, et al. A highly selective delta 1-opioid receptor antagonist: 7-benzylidenenaltrexone. Eur J Pharmacol. 1992;218(1):195-196. [Content Brief]
[2]. House RV, et al. Suppression of immune function by non-peptidic delta opioid receptor antagonists. Neurosci Lett. 1995 Sep 29;198(2):119-22. [Content Brief]
[3]. Miyata Y, et al. Opioid δ₁ receptor antagonist 7-benzylidenenaltrexone as an effective resistance reverser for chloroquine-resistant Plasmodium chabaudi. Bioorg Med Chem Lett. 2011 Aug 15;21(16):4710-2. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
BNTX maleate Related Classifications
HY-101307 Related Classifications
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