PD-161182
PD-161182 is a non-peptide NK-3 antagonist. PD-161182 can be studied in NK-3-related central nervous system disturbances, pain, inflammation, pulmonary and skin diseases.
For research use only. We do not sell to patients.
- CAS No.: 168570-35-2
- Formula: C29H40F2N4O4
- Molecular Weight:546.65
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CHO | IC50 |
1400 nM
Compound: 61
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Compound was tested for the inhibition of [125I]-[MePhe7]-NKB binding to cloned human Tachykinin receptor 3 in CHO cell lines
Compound was tested for the inhibition of [125I]-[MePhe7]-NKB binding to cloned human Tachykinin receptor 3 in CHO cell lines
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[PMID: 8648606] |
Chemical Information
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CAS No. 168570-35-2
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Molecular Weight 546.65
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Formula C29H40F2N4O4
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SMILES
O=C(N[C@](C)(C(NCCCCCCCNC(N)=O)=O)CC1=CC=CC(F)=C1F)O[C@@H](C(C)C)C2=CC=CC=C2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)