1198153-15-9
Chemical Structure
Epaminurad
Synonym(s): UR-1102; URC-102
- CAS. Nr.: 1198153-15-9
- Formula:C14H10Br2N2O3
- Molecular Weight:414.05
IUPAC Name: (3,5-dibromo-4-hydroxyphenyl)(2,3-dihydro-4H-pyrido[4,3-b][1,4]oxazin-4-yl)methanone
InChIKey: ZMVGQIIOXCGAFV-UHFFFAOYSA-N
SMILES: O=C(N1C2=C(OCC1)C=CN=C2)C3=CC(Br)=C(C(Br)=C3)O
Biological Activity: Epaminurad (UR-1102) is an orally active, potent and selective URAT1 (urate transporter 1) inhibitor, with a Ki of 0.057 μM. Epaminurad quite modestly inhibits OAT1 and OAT3 (organic anion transporter). Epaminurad is a uricosuric agent. Epaminurad can be used for gout and hyperuricemia research[1].
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Epaminurad | 99.75% | Epaminurad (UR-1102) is an orally active, potent and selective URAT1 (urate transporter 1) inhibitor, with a Ki of 0.057 μM. Epaminurad quite modestly inhibits OAT1 and OAT3 (organic anion transporter). Epaminurad is a uricosuric agent. Epaminurad can be used for gout and hyperuricemia research. | ||||||||||||||||||||
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Epaminurad (Standard) | ≥98% | Epaminurad (Standard) is the analytical standard of Epaminurad (HY-111345). This product is intended for research and analytical applications. Epaminurad (UR-1102) is an orally active, potent and selective URAT1 (urate transporter 1) inhibitor, with a Ki of 0.057 μM. Epaminurad quite modestly inhibits OAT1 and OAT3 (organic anion transporter). Epaminurad is a uricosuric agent. Epaminurad can be used for gout and hyperuricemia research. | ||||||||||||||||||||
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Similarity Score 0.98
HY-111345AEpaminurad hydrochloride -
Similarity Score 0.65
HY-101439JTT-552 -
Similarity Score 0.55
HY-126324IV-23 -
Similarity Score 0.54
HY-158194α2C adrenoceptor agonist 1 -
Similarity Score 0.53
HY-1191663,5,4'-Tribromosalicylanilide -
Similarity Score 0.52
HY-161674Monoamine Oxidase B inhibitor 4 -
Similarity Score 0.52
HY-184312PPAR agonist 8 -
Similarity Score 0.52
HY-110237BX430 -
Similarity Score 0.52
HY-175364Antiparasitic agent-27 -
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