181587-01-9
181587-01-9
Chemical Structure
Ethiprole
- CAS No.: 181587-01-9
- Formula:C13H9Cl2F3N4OS
- Molecular Weight:397.20
IUPAC Name: 5-amino-1-(2,6-dichloro-4-(trifluoromethyl)phenyl)-4-(ethylsulfinyl)-1H-pyrazole-3-carbonitrile
InChIKey: FNELVJVBIYMIMC-UHFFFAOYSA-N
SMILES: N#CC1=NN(C(N)=C1S(CC)=O)C2=C(C=C(C=C2Cl)C(F)(F)F)Cl
Biological Activity: Ethiprole is an insecticide.Metabolic sulfones are produced faster than Fipronil (HY-B0822) in CYP3A4-expressing cells and in vivo in mouse brain and liver.Ethiprole's sulfide, sulfoxide, sulfone and desulfinyl derivatives have better biological activity[1].
| Cat. No. | Nom du produit | Pureté | Description | Pricing | |||||||||||||||||||
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Ethiprole | 98.87% | Ethiprole is an insecticide.Metabolic sulfones are produced faster than Fipronil (HY-B0822) in CYP3A4-expressing cells and in vivo in mouse brain and liver.Ethiprole's sulfide, sulfoxide, sulfone and desulfinyl derivatives have better biological activity. | ||||||||||||||||||||
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Ethiprole (Standard) | ≥98% | Ethiprole (Standard) is the analytical standard of Ethiprole. This product is intended for research and analytical applications. Ethiprole is an insecticide.Metabolic sulfones are produced faster than Fipronil (HY-B0822) in CYP3A4-expressing cells and in vivo in mouse brain and liver.Ethiprole's sulfide, sulfoxide, sulfone and desulfinyl derivatives have better biological activity. | ||||||||||||||||||||
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Sisapronil | Sisapronil is a phenylpyrazole ectoparasiticide, that is widely used in the veterinary field. | |||||||||||||||||||||
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Flufiprole | Flufiprole is a nonsystemic phenylpyrazole insecticide targeting the GABA receptor used in the rice field. Flufiprole is excellent in controlling a wide range of pests. | |||||||||||||||||||||
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Fipronil sulfone | 99.85% | Fipronil sulfone is the major metabolite of Fipronil.Fipronil sulfone selectively inhibits |
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GABA-IN-2 | GABA-IN-2 (Compound 5) is a GABA inhibitor. GABA-IN-2 has larvicidal activity and insecticidal effect, with mortality rates of 87% at 50 mg/L. | |||||||||||||||||||||
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APS3 | APS3 is a GABA and nACh receptors inhibitor, with a LC50 of 7.2423 μg/mL against Plutella xylostella. | |||||||||||||||||||||
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M&B 39279 | M&B 39279 is an inhibitor of protoporphyrinogen oxidase (Protoporphyrinogen Oxidase). M&B 39279 induces protoporphyrin IX accumulation, light-dependent lipid peroxidation, degradation of membranes and organelles, and reduction of photosynthesis. M&B 39279 functions through the mechanism of action of diphenyl ether herbicides, and can be used for studies on PPO inhibition and herbicide mechanisms of action. | |||||||||||||||||||||
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Fipronil (Standard) | 99.49% | Fipronil (Standard) is the analytical standard of Fipronil. This product is intended for research and analytical applications. Fipronil is a broad-spectrum insecticide effective against Lepidoptera species as well as thrips, locusts, ants, cockroaches, fleas and ticks. Fipronil selectively inhibits GABA receptor with IC50s of 30 nM and 1600 nM for cockroach and rat GABA receptors, respectively. Glutamate-gated chloride channels (GluCls), which are present in cockroaches but not in mammals, are sensitive to the blocking effect of Fipronil. Fipronil also induces apoptosis in HepG2 cells and promotes the expression of CYP1A1 and CYP3A4 mRNA in human hepatocytes. | ||||||||||||||||||||
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Pyriprole | Pyriprole can be used against cat flea. Pyriprole disrupts the flea life cycle through killing of adult fleas before they lay eggs. Pyriprole has residual effect on debris from dog, which results in a decreased ability of cat flea larvae to complete development to the adult stage. | |||||||||||||||||||||
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Fipronil desulfinyl (Standard) | ≥98% | Fipronil desulfinyl (Standard) is the analytical standard of Fipronil desulfinyl. This product is intended for research and analytical applications. Fipronil desulfinyl is a photodegradation product of the insecticide Fipronil (HY-B0822) and has similar in vivo toxicity to Fipronil but higher environmental pollution. | ||||||||||||||||||||
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Fipronil sulfide | Fipronil sulfide is a toxic, persistent metabolite of Fipronil (HY-B0822). Fipronil is a broad-spectrum insecticide. | |||||||||||||||||||||
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