199864-87-4
199864-87-4
Chemical Structure
RS-127445
- CAS No.: 199864-87-4
- Formula:C17H16FN3
- Molecular Weight:281.33
IUPAC Name: 4-(4-fluoronaphthalen-1-yl)-6-isopropylpyrimidin-2-amine
InChIKey: ZZZQXCUPAJFVBN-UHFFFAOYSA-N
SMILES: NC1=NC(C(C)C)=CC(C2=C3C=CC=CC3=C(F)C=C2)=N1
Biological Activity: RS-127445 is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist with a pKi of 9.5. RS-127445 shows 1000 fold selectivity for this receptor as compared to numerous other receptor and ion channel binding sites[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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RS-127445 | 99.95% | RS-127445 is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist with a pKi of 9.5. RS-127445 shows 1000 fold selectivity for this receptor as compared to numerous other receptor and ion channel binding sites. | ||||||||||||||||||||
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References
Keywords
