254740-64-2
254740-64-2
Chemical Structure
Sparsentan
Synonym(s): RE-021; DARA-a
- CAS No.: 254740-64-2
- Formula:C32H40N4O5S
- Molecular Weight:592.75
IUPAC Name: 4'-((2-butyl-4-oxo-1,3-diazaspiro[4.4]non-1-en-3-yl)methyl)-N-(4,5-dimethylisoxazol-3-yl)-2'-(ethoxymethyl)-[1,1'-biphenyl]-2-sulfonamide
InChIKey: WRFHGDPIDHPWIQ-UHFFFAOYSA-N
SMILES: O=S(C1=CC=CC=C1C2=CC=C(CN3C(CCCC)=NC4(CCCC4)C3=O)C=C2COCC)(NC5=NOC(C)=C5C)=O
Biological Activity: Sparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Sparsentan | 99.87% | Sparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively. | ||||||||||||||||||||
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Sparsentan-d5 | Sparsentan-d5 is deuterium labeled Sparsentan. Sparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively. | |||||||||||||||||||||
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References
Keywords
