2810747-78-3
2810747-78-3
Chemical Structure
BLU0588
- CAS 番号: 2810747-78-3
- Formula:C26H25N5O
- Molecular Weight:423.51
InChIKey: YXSWSKFLTNJZEO-DNQXCXABSA-N
SMILES: O=C(C1=CN=C(C2=C3C(NC=C3)=NC=C2)C=C1)N[C@H]4[C@H](N5CCCC5)CC6=CC=CC=C64
Biological Activity: BLU0588 is an orally active, potent and selective PRKACA (protein kinase cAMP-activated catalytic subunit alpha) kinase inhibitor, with an IC50 of 1 nM and dissociation constant (Kd) of 4 nM. BLU0588 can be used for fibrolamellar carcinoma (FLC) research[1].
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BLU0588 | 97.63% | BLU0588 is an orally active, potent and selective PRKACA (protein kinase cAMP-activated catalytic subunit alpha) kinase inhibitor, with an IC50 of 1 nM and dissociation constant (Kd) of 4 nM. BLU0588 can be used for fibrolamellar carcinoma (FLC) research. | ||||||||||||||||||||
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References
Keywords
