52029-86-4
Chemical Structure
STO-609
- CAS No.: 52029-86-4
- Formula:C19H10N2O3
- Molecular Weight:314.29
IUPAC Name: 7-oxo-7H-benzo[de]benzo[4,5]imidazo[2,1-a]isoquinoline-3-carboxylic acid
InChIKey: MYKOWOGZBMOVBJ-UHFFFAOYSA-N
SMILES: O=C(C1=C2C3=C(C4=NC5=CC=CC=C5N4C(C3=CC=C2)=O)C=C1)O
Biological Activity: STO-609 is a selective and cell-permeable inhibitor of the Ca2+/calmodulin-dependent protein kinase kinase (CaM-KK), with Ki values of 80 and 15 ng/mL for recombinant CaM-KKα and CaM-KKβ, respectively. STO-609 inhibits AMP-activated protein kinase kinase (AMPKK) activity in HeLa cell lysates with an IC50 ~0.02 g/ml.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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STO-609 | 98.20% | STO-609 is a selective and cell-permeable inhibitor of the Ca2+/calmodulin-dependent protein kinase kinase (CaM-KK), with Ki values of 80 and 15 ng/mL for recombinant CaM-KKα and CaM-KKβ, respectively. STO-609 inhibits AMP-activated protein kinase kinase (AMPKK) activity in HeLa cell lysates with an IC50 ~0.02 g/ml. | ||||||||||||||||||||
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Keywords
